Cytochrome P450 substrates
Injected separately or as a cocktail to assess CYP450 isoform activities
Drug CYP450
Caffeine CYP1A2
Chlorzoxazone CYP2E1
Dextromethorphan CYP2D6
Diclofenac CYP2C9
Esomeprazole CYP2C19
Metoprolol CYP2D6
Midazolam CYP3A4
Theophylline CYP1A2
Tolbutamide CYP2C9
Other Drugs
Aripiprazole
Brimonidine
Bupivacaine
Famotidine Organic cation transporter substrate
Fentanyl
Glyburide
Levetiracetam
Memantine
Minocycline
Phenytoin
Probenecid Organic anion transporter substrate
Propofol
New procedures are constantly being developed. Please Contact Us for more information.